Product Overview
4 hour antihistamine allergy tablets that relieves sneezing, runny nose, itchy, watery eyes, and itchy throat.
Major Chlorpheniramine Maleate 4 mg - 100 Tablets | Chlor-Trimeton
- 4 hour allergy tablets
- Antihistamine
- Relieves sneezing, runny nose, itchy, watery eyes, itchy throat
Expiration Date: 8-2026
Ingredients
- Active: Chlorpheniramine Maleate 4 mg - Antihistamine
- Inactive: Corn Starch, D&C Yellow #10 Aluminum Lake, Lactose Anhydrous, Magnesium Stearate, Microcrystalline Cellulose
Uses
- Temporarily relieves these symptoms due to hay fever or other respiratory allergies:
- Sneezing
- Runny nose
- Itchy, watery eyes
- Itching of the nose
FULL DESCRIPTION
Drug Facts
Active Ingredients
- Chlorpheniramine Maleate - 4 mg
- Purpose: Antihistamine
Uses
- Temporarily relieves these symptoms due to hay fever or other respiratory allergies:
- Sneezing
- Runny nose
- Itchy, watery eyes
- Itching of the nose
Warnings
- Do Not Use
- To make a child sleepy
- Ask a Doctor Before Use if You Have
- A breathing problem such as emphysema or chronic bronchitis
- Glaucoma
- Difficulty in urination due to enlargement of the prostate gland
- Ask a Doctor or Pharmacist Before Use if You Are
- Taking sedatives or tranquilizers
- When Using This Product
- Drowsiness may occur
- Avoid Alcoholic beverages
- Excitability may occur especially in children
- Use caution when driving a motor vehicle or operating machinery
- Alcohol, sedatives, and tranquilizers may increase drowsiness
- If Pregnant or Breast-Feeding
- Ask a health professional before use
- Keep Out of Reach of Children
- In case of overdose, get medical help or contact a Poison Control Center
Directions
- Take every 4 to 6 hours, or as directed by a doctor
- Adults and Children 12 Years and Over
- 1 tablet
- Do not exceed 6 tablets in 24 hours
- Children 6 to Under 12 Years
- 1/2 tablet (break tablet in half)
- Do not exceed 3 whole tablets in 24 hours
- Children Under 6 Years
- Do not use
Other Information
- Store at 25ºC
- Excursions permitted between 15ºC-30ºC (59ºF-86ºF)
- Protect from excessive moisture
- See end flap for expiration date and lot number
Inactive Ingredients
- Corn Starch, D&C Yellow #10 Aluminum Lake, Lactose Anhydrous, Magnesium Stearate, Microcrystalline Cellulose
Is chlorpheniramine maleate a strong antihistamine?
Yes, chlorpheniramine maleate is considered a strong antihistamine. It belongs to a class of medications known as first-generation antihistamines. Chlorpheniramine maleate is used to relieve symptoms associated with allergic conditions such as hay fever, allergic rhinitis, and hives.
As a strong antihistamine, chlorpheniramine maleate has potent anticholinergic effects, meaning it can cause sedation and drowsiness. It is known to have a significant impact on the central nervous system, leading to a sedating effect that can make individuals feel sleepy or groggy. Consequently, chlorpheniramine maleate is often included in over-the-counter medications designed specifically for nighttime use to help with sleep.
However, due to its sedating properties, chlorpheniramine maleate may not be suitable for everyone, especially those who need to remain alert or engage in activities that require mental alertness. Additionally, it is important to follow the recommended dosage and usage instructions provided by a healthcare professional or on the medication packaging to ensure safe and effective use. Consulting a healthcare provider or pharmacist is always advisable before starting any new medication.
What is chlorpheniramine maleate used for?
Chlorpheniramine maleate is an antihistamine medication that is used to relieve symptoms associated with various allergic conditions, including:
1. Allergic rhinitis: It helps alleviate symptoms such as sneezing, runny or itchy nose, and nasal congestion caused by allergies to substances like pollen, dust mites, or pet dander.
2. Hay fever: Chlorpheniramine maleate can provide relief from symptoms such as sneezing, itching, watery eyes, and nasal congestion that occur during the pollen season.
3. Allergic conjunctivitis: It can help reduce itching, redness, and watering of the eyes caused by allergies.
4. Hives (urticaria): Chlorpheniramine maleate is sometimes used to alleviate itching and reduce the appearance of hives caused by allergic reactions.
It is important to note that chlorpheniramine maleate is typically used for short-term symptomatic relief of allergic symptoms and is not meant for long-term use. The specific dosage and usage instructions may vary depending on the formulation, brand, and individual factors, so it is advisable to follow the directions provided by a healthcare professional or on the medication packaging. If you have any specific concerns or questions about the use of chlorpheniramine maleate, it's best to consult a healthcare provider.
Is chlorpheniramine maleate the same as Zyrtec?
No, chlorpheniramine maleate and Zyrtec (generic name: cetirizine) are different medications. While both are antihistamines used to relieve allergy symptoms, they belong to different classes of antihistamines and have different active ingredients.
Chlorpheniramine maleate is a first-generation antihistamine, known for its sedating properties. It has been used for many years to treat allergic conditions like allergic rhinitis, hay fever, and hives. It is available in various over-the-counter and prescription formulations.
On the other hand, Zyrtec (cetirizine) is a second-generation antihistamine. It is also used to relieve symptoms of allergic conditions such as hay fever, allergic rhinitis, and hives. Compared to first-generation antihistamines like chlorpheniramine, cetirizine is generally less sedating and is often preferred for its non-drowsy effect. Zyrtec is available over-the-counter in many countries and also comes in prescription-strength formulations.
While both medications work by blocking the effects of histamine, they have different chemical structures and may have varying degrees of effectiveness and side effects for different individuals. It's important to consult a healthcare professional or pharmacist to determine which medication is most suitable for your specific needs.
What is the disadvantage of chlorpheniramine?
Chlorpheniramine is an antihistamine medication commonly used to relieve symptoms of allergies, such as sneezing, itching, watery eyes, and runny nose. While it is generally considered safe and effective, there are a few potential disadvantages or side effects associated with its use. These include:
1. Sedation: Chlorpheniramine can cause drowsiness and sedation. This effect may impair cognitive function and alertness, making activities such as driving or operating heavy machinery dangerous. It is important to be cautious when taking chlorpheniramine, especially when engaging in activities that require mental alertness.
2. Dry mouth and blurred vision: Chlorpheniramine can cause dryness of the mouth, throat, and nasal passages, leading to discomfort. It may also cause blurred vision or difficulty focusing due to its anticholinergic effects.
3. Urinary retention: Chlorpheniramine can sometimes affect the urinary system, causing difficulty or discomfort in passing urine. This is more likely to occur in individuals with underlying prostate enlargement or bladder conditions.
4. Increased heart rate: In some cases, chlorpheniramine can lead to an increased heart rate or palpitations. This effect is more likely to occur at higher doses or in individuals with pre-existing heart conditions.
5. Interactions with other medications: Chlorpheniramine may interact with certain medications, including central nervous system depressants, such as alcohol, sedatives, or tranquilizers. These interactions can potentiate the sedative effects and increase the risk of adverse effects.
It's important to note that individual responses to medications can vary, and not everyone will experience these side effects. It is always recommended to consult a healthcare professional or pharmacist before starting any new medication to discuss potential risks, interactions, and alternative options.
What is the OTC brand name for chlorpheniramine?
One common over-the-counter (OTC) brand name for chlorpheniramine is Chlor-Trimeton. Chlor-Trimeton contains chlorpheniramine as its active ingredient and is available in various forms, such as tablets, capsules, or liquid formulations. However, it's important to note that the availability of specific brands may vary depending on the country or region. It is always recommended to check with local pharmacies or retailers for the specific OTC brand names available in your area.
How strong is chlorphenamine?
The strength of chlorpheniramine, also known as chlorphenamine, can vary depending on the formulation and dosage form. Chlorpheniramine is available in different strengths, typically ranging from 2 mg to 4 mg per tablet or capsule. The liquid formulations may have varying concentrations as well.
When using over-the-counter (OTC) chlorpheniramine products, it is important to carefully read and follow the instructions on the packaging and consult with a healthcare professional or pharmacist if you have any questions or concerns. They can provide guidance on the appropriate dosage and strength based on your specific needs and medical history.
Is chlorpheniramine maleate stronger than loratadine?
Chlorpheniramine maleate and loratadine are both antihistamine medications, but they have different potency and characteristics. In general, chlorpheniramine maleate is considered to have a stronger sedative effect compared to loratadine.
Chlorpheniramine is a first-generation antihistamine that has a stronger tendency to cause sedation and drowsiness. It can cross the blood-brain barrier more easily, leading to its sedative effects. This sedation can be beneficial for individuals who experience difficulty sleeping due to allergies or cold symptoms. However, it can also be a disadvantage for those who need to remain alert and focused during the day.
On the other hand, loratadine is a second-generation antihistamine that is less likely to cause sedation. It is designed to be less sedating and have a longer duration of action compared to first-generation antihistamines like chlorpheniramine. Loratadine is often preferred for daytime use, as it is less likely to cause drowsiness and allows individuals to remain more alert and functional.
It's important to note that individual responses to medications can vary, and some individuals may still experience drowsiness or other side effects with loratadine. It's always advisable to follow the recommended dosages and consult with a healthcare professional or pharmacist for personalized advice based on your specific needs and medical history.
Which is better chlorpheniramine maleate or diphenhydramine?
The choice between chlorpheniramine maleate and diphenhydramine depends on various factors, including the specific symptoms being treated and individual response to the medications. Both chlorpheniramine maleate and diphenhydramine are first-generation antihistamines and have similar mechanisms of action, but they have some differences in their characteristics:
1. Sedation: Both chlorpheniramine maleate and diphenhydramine can cause sedation and drowsiness. However, diphenhydramine is generally considered to have a stronger sedative effect compared to chlorpheniramine. Diphenhydramine is often used as a sleep aid due to its sedating properties, while chlorpheniramine may have a milder sedative effect.
2. Duration of action: Chlorpheniramine has a shorter duration of action, typically lasting around 4 to 6 hours, whereas diphenhydramine has a longer duration of action, typically lasting around 6 to 8 hours. The longer duration of action of diphenhydramine can be beneficial for individuals who need symptom relief throughout the night.
3. Side effects: Both medications can cause common side effects such as dry mouth, blurred vision, and urinary retention. Diphenhydramine may have a higher incidence of these side effects compared to chlorpheniramine.
4. Drug interactions: Both chlorpheniramine and diphenhydramine can interact with other medications, especially those with sedative effects. It's important to check for potential drug interactions with other medications you may be taking.
The choice between chlorpheniramine maleate and diphenhydramine should be based on the individual's symptoms, desired level of sedation, and other factors such as the need for daytime functionality or the duration of action required. It is recommended to consult with a healthcare professional or pharmacist to determine the most suitable option based on your specific needs and medical history.
Can you take Benadryl with chlorpheniramine maleate?
Taking Benadryl (diphenhydramine) and chlorpheniramine maleate together is generally not recommended without consulting a healthcare professional. Both medications are first-generation antihistamines that have sedating effects. Combining them can potentially increase the risk of excessive sedation and other side effects.
Taking multiple antihistamines simultaneously may also lead to an increased risk of anticholinergic side effects, such as dry mouth, blurred vision, constipation, and urinary retention. Additionally, both diphenhydramine and chlorpheniramine can interact with other medications, so it's important to consider any potential drug interactions.
If you need relief from allergy symptoms or other conditions, it is best to consult with a healthcare professional or pharmacist. They can provide guidance on the appropriate medications, dosages, and potential interactions based on your specific needs and medical history.
What is chlorpheniramine maleate comparable to?
Chlorpheniramine maleate is comparable to other first-generation antihistamines, such as diphenhydramine (Benadryl) and brompheniramine. These medications belong to the same class of antihistamines and have similar mechanisms of action. They are used to relieve symptoms of allergies, such as sneezing, itching, watery eyes, and runny nose.
While chlorpheniramine, diphenhydramine, and brompheniramine have some differences in terms of their potency, duration of action, and sedative effects, they are generally considered to be comparable in terms of their effectiveness in treating allergy symptoms. However, individual responses to these medications can vary, and some people may find one medication more effective or better tolerated than others.
It's important to note that there are also second-generation antihistamines available, such as loratadine (Claritin), cetirizine (Zyrtec), and fexofenadine (Allegra). These medications are generally preferred for their non-sedating properties and longer duration of action, making them suitable for daytime use. If you are considering antihistamine options, it's recommended to consult with a healthcare professional or pharmacist who can recommend the most suitable medication based on your specific needs and medical history.
Which antihistamine is the most effective?
There are several antihistamines available on the market, and the effectiveness of each can vary depending on individual factors and specific symptoms.
First-generation antihistamines, such as diphenhydramine (Benadryl) and chlorpheniramine (Chlor-Trimeton), are effective in relieving symptoms like itching, sneezing, and runny nose. However, they are known to cause drowsiness and may not be ideal for daytime use.
Second-generation antihistamines, such as cetirizine (Zyrtec), loratadine (Claritin), and fexofenadine (Allegra), are often preferred due to their non-drowsy formulations. These antihistamines are effective in treating allergy symptoms and are usually recommended for regular use.
The choice of the most effective antihistamine depends on individual factors, such as the specific allergy symptoms, personal response to the medication, and any other existing medical conditions or medications being taken. It is best to consult with a healthcare professional, such as a doctor or pharmacist, who can consider your specific situation and provide appropriate recommendations.
